1 natijalarini 12-20 Ko'rsatilgan

CAS NO. MAHSULOT NOMI Umumiy
    1351522-04-7 AC710 (1351522-04-7)

    AC710 kuchli potentsial, og'izdan faol va selektiv trombotsitlar bilan o'sish omili retseptorlari-oilaviy kinaz inhibitori bo'lib, potentsial qarshi ta'sirga ega.

    1002304-34-8 AMG208 (1002304-34-8)

    AMG 208 - epiteliya yuzasida ifodalangan yaxshi tavsiflovchi rezektsion tirozin kinaz bo'lgan c-Metning kichik molekula inhibitori.

    883986-34-8 AZD2932 (883986-34-8)

    AZD2932 50 nM, 8 nM, 4 nM va VEGFR-7, PDGFRb, Flt-9, 2 nM uchun IC3 bilan kuchli va mutil maqsadli protein tirozin kinaz inhibitori.

    1265229-25-1 CH-5183284 (1265229-25-1)

    CH5183284 50 nM, 9.3 nM, 7.6 nM, va FGFR22, FGFR290, FGFR1 va FGFR uchun 2 nM IC3 bilan tanlangan va og'zaki mavjud bo'lgan FGFR inhibitori ...

    343787-29-1 CP-673451 (343787-29-1)

    CP-673451 hujayra-bo'lmagan tekshiruvlarda 50 nM / 10 nM ning IC1 bilan PDGFRa / b ni selektiv inhibitori bo'lib, boshqa angijalar bo'yicha 450-qatlamliligi ...

    405169-16-6 Dovitinib (TKI-258) (405169-16-6)

    Dovitinib (TKI258, CHIR258) 3 nM / 50 nM ning IC1 bilan sinfi kuchli, ko'pincha sinf III (FLT2 / c-Kit) uchun multitgetgeted RTK inhibitoridir ...

    1058137-23-7 E-3810 (1058137-23-7)

    E-3810 VEGF va FGF retseptorlari kuchli va tanlangan er-xotin inhibitori bo'lib, VEG uchun 50 nM, 7 nM, 25 nM, 10 nM va 17.5 nM ning IC82.5 qiymatlari bilan ...

    1100598-32-0 EMD1214063 (1100598-32-0)

    EMD1214063 potentsial antineoplastik faollik bilan MET tirozin kinaz inhibitori. EMd 1214063 selektiv tirozin kinaz inhibitori ...

    1708971-72-5 FGFR4-IN-1 (1708971-72-5)

    FGFR4-IN-1 kuchli va tanlangan FGFR4 inhibitori. FGFR4 gastrik saraton uchun yangi terapevtik maqsad bo'lishi mumkin. FGFR4-IN-1 muhim darajada ...

    1254473-64-7 LY2874455 (1254473-64-7)

    LY2874455 50 nM, 2.8 nM, 2.6 nM va 6.4 nM bilan FGFR6, FGFR1, FGFR2 va FGFR3 uchun IC4 bilan pan-FGFR inhibitori va shuningdek, ...

    790299-79-5 Masitinib (AB1010) (790299-79-5)

    Masitinib (AB1010) hayvonlarda mast hujayralari o'smalarini, ayniqsa, itlarni davolashda ishlatiladigan tirozin-kinaz inhibitoridir. Kirish boshlanganidan beri ...

    366017-09-6 Mubritinib (TAK 165) (366017-09-6)

    TAK-165 sifatida ham tanilgan Mubritinib, Takeda tomonidan saratonni davolashda ishlab chiqilgan bir protein kinaz inhibitori. To'liq ...