1 natijalarini 12-630 Ko'rsatilgan

CAS NO. MAHSULOT NOMI Umumiy
    856925-71-8 (-) - Blebbistatin (856925-71-8)

    (-) - Blebbistatin nekrozsiz miyosin II ATPaz uchun xNUMXmX dan IC50 bilan hujayra-o'tkazuvchan inhibitordir, myozinning engil zanjirli kinazini inhibe qilmaydi ...

    1268524-70-4 (+) - JQ1 (1268524-70-4)

    (+) - JQ1 - BET bromodomain inhibitori, BRD50 (77 / 33) uchun 4 nM / 1 nM ning IC2 bilan, BET oilasining barcha bromodomenleriga bog`langan, ammo bromga emas.

    5142-23-4 3-Methyladenine (3-MA) (5142-23-4)

    3-Metiladenin III-fosfatidilinositol 3-kinaz (PI 3-kinaz) ning inhibitori hisoblanadi .Cerebellar granül hujayralarini apoptozdan himoya qilish mumkin ...

    1668553-26-1 A-1210477 (1668553-26-1)

    A-1210477 Ki va IC1 ning 50 nM va 0.454 nM bilan mos keladigan kuchli va tanlangan MCL-26.2 inhibitori bo'lib, u 100-kattalikdagi ...

    1527503-11-2 A-366 (1527503-11-2)

    A-366 kuchli va tanlangan G9a / GLP histon lizin metiltransferaza inhibitori (ICx = 3.3 nM). 1000-qavat uchun tanlanganligini ko'rsatadi ...

    552325-73-2 A-674563 (552325-73-2)

    A-674563 1nM ning IC50 qiymatiga ega potentsial, og'zaki ravishda mavjud Akt11 inhibitori. Shuningdek, ICA2 qiymati bilan PKA va CDK50ga qarshi faoliyat ko'rsatiladi ...

    844499-71-4 A-769662 (844499-71-4)

    A-769662 50 mM.A-0.8 ning EC769662 bilan kuchli, qaytariladigan AMP faollashtirilgan oqsil kinozasi (AMPK) faollashtiruvchisi bo'lib, b ...

    934162-61-5 A-966492 (934162-61-5)

    A-966492 PARP1 va PARP2 ning yangi va kuchli inhibitori bo'lib, Ki ning 1 nM va 1.5 nM bilan navbati bilan.

    1166227-08-2 A66 (1166227-08-2)

    A66 110 nM ning IC50 bilan juda aniq va tanlangan p32a inhibitoridir, boshqa sinf-I PI100K izoformiga nisbatan p110a uchun 3 marta sayrlilik ...

    607737-87-1 A77-01 (607737-87-1)

    77-01 kuchli TGF-RRI (ALK-5) inhibitori (IC50 = 34 nM). TGF-b transkripsiyadan foydalanishni inhibe qiladi. TGF-b induktsiyasining proliferatsiyasini inhibe ...

    909910-43-6 A83-01 (909910-43-6)

    A 83-01 - TGF-b I I retseptorlari ALK5 kinazining kuchli inhibitori, ALK4 turi I ning aktiv / nodal retseptorlari va ALK7 tipidagi I nodal retseptorlari.

    714971-09-2 AC480 (BMS-599626) (714971-09-2)

    BMS-480 deb nomlanuvchi AC599626 raklar, metastazlar va HER2 yoki EGFR Expressing Advanced So ...

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